Template:Glucocorticoid activity of selected steroids in vitro

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Glucocorticoid activity of selected steroids in vitro

Steroid Class TR ()a GR (%)b
Template:No selflink Corticosteroid ++ 100
Template:No selflink Estrogen 0
Template:No selflink Progestin + 14
Template:No selflink Progestin + 27
Template:No selflink Progestin 1
Template:No selflink Progestin + 29
Template:No selflink Progestin 0
Template:No selflink Progestin 1
Template:No selflink Progestogen + 10
Footnotes: a = Thrombin receptor (TR) upregulation (↑) in vascular smooth muscle cells (VSMCs). b = RBA (%) for the glucocorticoid receptor (GR). Strength: – = No effect. + = Pronounced effect. ++ = Strong effect. Sources: [1]

References

  1. Kuhl H (2005). "Pharmacology of estrogens and progestogens: influence of different routes of administration" (PDF). Climacteric. 8 Suppl 1: 3–63. doi:10.1080/13697130500148875. PMID 16112947. S2CID 24616324.