Template:Affinities of dydrogesterone and related steroids

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Affinities of dydrogesterone and related steroids

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Progestogen PR AR GR ERα
Ki (nM) RBA (%) Ki (nM) RBA (%) Ki (nM) RBA (%) Ki (nM)
Template:No selflink 125.9 15.9 251.2 10.0 361.2 17.5 >10,000
Template:No selflink 125.9 15.9 3162.3 0.8 3162.3 2.0 >10,000
Template:No selflink 20.0 100 25.1 100 63.1 100 >10,000
Sources: [1]
Template documentation

References

  1. Rižner TL, Brožič P, Doucette C, Turek-Etienne T, Müller-Vieira U, Sonneveld E, van der Burg B, Böcker C, Husen B (May 2011). "Selectivity and potency of the retroprogesterone dydrogesterone in vitro". Steroids. 76 (6): 607–15. doi:10.1016/j.steroids.2011.02.043. PMID 21376746.